Formulation | Lopinavir+ritonavir (mg/mL) | Composition | (glycerol) |
A1 | 16.0+4.0 | Phase 1: ethanol 2 mL, glycerol 1.6 mL; phase 2: water 22 mL | 6% |
A2 | 14.9+3.7 | Phase 1: ethanol 2 mL, glycerol 3 mL; phase 2: water 21.8 mL | 11% |
A3 | 14.3+3.6 | Phase 1: ethanol 2 mL, glycerol 4.2 mL; phase 2: water 21.8 mL | 15% |
A4* | 14.9+3.7 | Phase 1: ethanol 2 mL, glycerol 3 mL; phase 2: water 21.8 mL | 11% |
B1 | 14.3+3.6 | Ethanol 2 mL, glycerol 3 mL, water 23 mL | 11% |
B2 | 14.3+3.6 | Water 28 mL | – |
*Coating film removed from tablets.